Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04669
Ion Channel
Potassium channel subfamily K member 3
Peptide Function
Inhibitor
Gene Name
KCNK4
Activity Data (nM)
IC50
80 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
CSCSSLMDKECVYFCHLDIIW
Peptide UniProt Accession
Not available
UniParc
UPI000002E63D
Peptide Synonyms/Alias
[Endothelin-1; ET-1; Endothelin I; 123626-67-5; CHEMBL3775234; 1-(4-Hydroxyphenyl)-2;4;6-triphenylpyridinium hydroxide inner salt hydrate; GTPL989; BDBM50155246; Endothelin 1; >=97.0% (HPLC); Endothelin 1; >=97% (HPLC); powder; Endothelin 1??; Vetec(TM) reagent grade; >=97%; L-cysteinyl-L-seryl-L-cysteinyl-L-seryl-L-seryl-L-leucyl-L-methionyl-L-alpha-aspartyl-L-lysyl-L-alpha-glutamyl-L-cysteinyl-L-valyl-L-tyrosyl-L-phenylalanyl-L-cysteinyl-L-histidyl-L-leucyl-L-alpha-aspartyl-L-isoleucyl-L-isoleucyl-L-tryptophan (1->15);(3->11)-bis(disulfide)]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
123626-67-5
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−80 mV
Temperature
Room Temperature
Test Method
Patch-clamping
Test Species
Not specified
Binding Information
Binding Site
Transmembrane domain
Binding Site Residue
Ser(393)
Ion Channel Information
Gene Abbreviation (ABB)
K2P
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available